WebA series of MMP-1 inhibitors have been identified based upon a Methyl rosmarinate scaffold using structure-based drug design methods. The best compound in the series showed an IC50 value of 0.4 muM. A docking … WebDownload scientific diagram H-NMR and 13 C-NMR data and NOESY correlations of the diterpene 1 and derivatives 2a and 2b (400 and 100 MHz, respectively; CDCl 3 ; δ-values). from publication: The ...
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WebApr 3, 2024 · Thammason, H., Khetkam, P., Pabuprapap, W., Suksamrarn, A., & Kunthalert, D. (2024). Ethyl rosmarinate inhibits lipopolysaccharide-induced nitric oxide and ... WebDescription. Ursolic acid, a naturally occurring triterpenoid, induces the apoptosis of human cancer cells through multiple signaling pathways. Ursonic acid has antiviral activity against Herpes simplex virus types I and II in vitro; it also could be used in preparation of depression treatment medicine. Targets.
Webethyl rosmarinate 抑制酪氨酸酶、α-葡萄糖苷酶和基质金属蛋白酶-1 (MMP-1) 的活性。 产品描述 Methyl rosmarinate inhibit the activity of tyrosinase, α-glucosidase, and matrix metalloproteinase-1 (MMP-1).
WebButyl Rosmarinate. CHEMBL2335275. Molecular Weight: 416.4. Dates: Modify . 2024-01-28. Create . 2006-11-20. Butyl Rosmarinate is a natural product found in Isodon oresbius with data available. LOTUS - the natural products occurrence database. Contents. 1 Structures Expand this section. WebDec 19, 2024 · Ethyl rosmarinate (RAE) is one of the active constituents from Clinopodium chinense (Benth.) O. Kuntze, which is used for diabetic treatment in Chinese folk medicine. In this study, we ...
WebDec 19, 2024 · Ethyl rosmarinate (RAE) is one of the active constituents from Clinopodium chinense (Benth.) O. Kuntze, which is used for diabetic treatment in Chinese folk medicine. In this study, we investigated the protective effect of RAE on high glucose-induced injury in endothelial cells and explored its underlying mechanisms. Our results showed that both …
WebSep 28, 2024 · American ginseng (AG), the underground part of Panax quinquefolium L., is composed of four morphological regions, including main root (MR), lateral root (LR), fibrous root (FR), and rhizome (RH). In the … map of india 1930WebApr 1, 2024 · Turpesteryl ester (1), a new steroid, has been isolated from the ethyl acetate-soluble subfraction of the methanolic extract of Ipomoea turpethum (L.) R.Br., along with stigmasterol, β-sitostenone, rosmarinic acid, and methyl rosmarinate, reported for the first time from this species. Their structures were elucidated with the help of spectroscopic … map of india 1970WebDec 15, 2024 · of 73 mg of ethyl rosmarinate and 80 mg of propyl rosmarinate were obtained after the. Plants 2024, 10, 2773 9 of 21. reaction solutions were centrifuged, filtered, and evaporated. map of india 2011WebDec 19, 2024 · Ethyl rosmarinate (RAE) is an active component in CC with α-glucosidase inhibition and cytoprotection . It has been reported that RAE exhibited the most potent inhibitory effect on NO production in lipopolysaccharide-induced murine alveolar macrophage cells [ 17 ], and RAE induced relaxation in aortic rings via an endothelium … kroger pharmacy bellefontaine hoursWebJan 23, 2024 · Aiming at assessing the therapeutic effect of ethyl rosmarinate (ER) on ulcerative colitis (UC), the following activities were performed in vitro and in vivo in the present study. Firstly, a lipopolysaccharide (LPS)-induced RAW264.7 cell inflammation model was established to determine the level of inflammatory factors. Then, a UC mice … map of india 1956WebApr 3, 2024 · Ethyl rosmarinate inhibits lipopolysaccharide-induced nitric oxide and prostaglandin E 2 production in alveolar macrophages. European Journal of Pharmacology, 824, 17–23. doi:10.1016/j.ejphar.2024.01.042 kroger pharmacy beechmont avenueWebA series of MMP-1 inhibitors have been identified based upon a Methyl rosmarinate scaffold using structure-based drug design methods. The best compound in the series showed an IC50 value of 0.4 muM. A docking study was conducted for compound (S)-10n in order to investigate its binding interactions with MMP-1. map of india 1948